Deisgn of Benzoxathiazin old pub5

Design of benzoxathiazin-3-one 1,1-dioxides as a new class of irreversible serine hydrolase inhibitors: discovery of a uniquely selective PNPLA4 inhibitor

Publication Year: 2017
Kornahrens, A, Cognetta, A Brody D, Matthews ML, Cravatt BF & Boger D.
[PDF]  [External Link]

Kornahrens, A, Cognetta, A Brody D, Matthews ML, Cravatt BF & Boger D.. Design of benzoxathiazin-3-one 1,1-dioxides as a new class of irreversible serine hydrolase inhibitors: discovery of a uniquely selective PNPLA4 inhibitor. J. Am. Chem. Soc.  139, 7052–7061 (2017)